Electrochemical synthesis of hemiaminal from protected amino acids: A facile alternative way to access pro-drugs and ADC linkers via decarboxylative hydroxylation
Publication: Elsevier
Future of Medicine: How Small Molecules and Biologics Complement Each Other – A Medicinal Chemist’s Perspective
Publication: ACS Publication
Lead Optimization of a Pyrrole-Based Dihydroorotate
Publication: Journal of Medicinal Chemistry
Palladium‐Catalyzed Reductive Carbonylation of (Hetero) Aryl Halides and Triflates Using Cobalt Carbonyl as CO Source
Publication: Europen Journal of Organic Chemistry
Selective recruitment of γδ T cells by a bispecific antibody for the treatment of acute myeloid leukemia
Publication: Leukemia
US FDA approved drugs from 2015-June 2020-A perspective
Publication: Journal of Medicinal Chemistry
Potent antimalarials with development potential identified by structure-guided computational optimization of a pyrrole-based dihydroorotate dehydrogenase inhibitor series
Publication: Journal of Medicinal Chemistry
Structure-Based Optimization and Discovery of M3258, a Specific Inhibitor of the Immunoproteasome Subunit LMP7 (β5i)
Publication: Journal of Medicinal Chemistry
TNB-738, a biparatopic antibody, boosts intracellular NAD+ by inhibiting CD38 ecto-enzyme activity
Publication: mAbs
Systematic mutational analysis reveals an essential role of N275 in IgE stability
Publication: Biotechnology and Bioengineering, Wiley